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REFERAT NSAID
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REFERAT NSAID
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LEMBAR PENGESAHAN Obat Anti Jamur Sistemik
Referat Farmasi
Oleh:
HELVIANSYAH EL FARIZQI
2016.0.2.00!"
HENRY S#RYA$I %IRYA&AR'A2016.0.2.00!( ILIYIN SYAHAR FARIHA'#N NISA
2016.0.2.00"0
I)A)S#'RISNO
2016.0.2.00"1
I)ROA'#SSAQIYAH
2016.0.2.00"2
IN$IRA FIR$HA SYAFI'RI
2016.0.2.00"*
IN$IRA YO+AN'ARI RA,H)I
2016.0.2.00"
$iset--i /a /iterima seaai salah sat- t-as 3e4aiteraa 3lii3 5aia Farmasi RSAL $r. Ramela S-raaa Fa3-ltas &e/73tera Hat-ah S-raaa
S-raaa8 22 9-i 2016 )eetah-i8 $73ter 4emimi
BAB 1 PENDAHULUAN
1.1.
Latar Belakang
asie /ata 3e eraai 4-sat 4elaaa 3esehata seaia esar /ea 3el-ha eri. eatala3saaa 3as-s eri mem-t-h3a 4emahama a3a 4r7ses 4at7fisi7l7i eri ter-tama eri a mei3-ti s-at- 4r7ses iflamasi. 5eraai m7/alitas terse/ia /alam 4eaaa 3as-s eri am- 4a/a eri m7/alitas 4ertama a iasaa /i-a3a /alam 4eaaa eri a/alah 7at 7l7a 774iat ait- N7 Ster7i/al Ati;iflammat7r $r-s
ara 3imia. %ala-4- /emi3ia 7at;7at ii terata memili3i aa3 4ersamaa /alam efe3 tera4i ma-4- efe3 sam4i. r7t7ti4 7at 7l7a ii a/alah as4iri8 3area it- 7at 7l7a ii seri /ise-t -a seaai 7at miri4 as4iri (aspirin-like drugs).
1..
!u"uan P enelitian
#t-3 meetah-i efe3tifitas /a 3eamaa 7at NSAI$.
BAB !#NJAUAN PUS!A$A
.1.
!in"auan !entang N SA#D
.1.1. De%inisi NSA#D
Oat atiiflamasi
.1.. Mekanisme $e r"a NSA #D
Seaia esar efe3 tera4i /a efe3 sam4i NSAI$ er/asar3a atas 4ehamata i7sitesis 4r7stala/i <+=. a/a saat sel mealami 3er-sa3a8 ma3a a3a /ile4as3a eera4a me/iat7r 3imia. $i atara me/iat7r iflamasi8
4r7stala/i a/alah me/iat7r /ea 4era ter4eti. Eim a /ile4as3a saat a/a rasa me3ai3 ma-4- 3imia a/alah 4r7stala/i e/74er73si/a sitase <+HS= ata- si3l7 73siease <,OB= a memili3i /-a sisi 3ataliti3. Sisi a 4ertama a/alah sisi a3tif si3l7 73siease8 a a3a me-ah asam ara3hi/7at mea/i e/74er73si/ ++2. Sisi a laia a/alah sisi a3tif 4er73si/ase8 a a3a me-ah ++2 mea/i e/74er73si/ lai ait- +H2. +H2 sela-ta a3a /i4r7ses memet-3 +s8 4r7stasi3li /a tr7m73sa A28 a 3etiaa mer-4a3a me/iat7r -tama 4r7ses iflamasi. ,OB ter/iri atas /-a is7f7rm ait- ,OB;1 /a ,OB;2. +7l7a 7at ii mehamat eim si3l7 73siease <,OB= sehia 37Cersi asam ara3hi/7at mea/i ++2 tera-. Setia4 7at mehamat /ea >ara ere/a. &h-s-s 4arasetam7l8 hamata i7sitesis 4r7stala/i haa tera/i ila li3-aa re/ah 3a/ar 4er73si/a se4erti /i hi47talam-s. L73asi iflamasi iasaa mea/- aa3 4er73si/a a /ihasil3a 7leh le-37sit. Ii meelas3a mea4a efe3 ati iflamasi 4arasetam7l 4ra3tis ti/a3 a/a. Ihiisi i7sitesis 4r7stala/i 7leh as4iri meea3a asetilasi a irreCersiel /i sisi a3tif si3l7 73iease8 se/a3a sisi a3tif 4er73si/ase ti/a3 ter4ear-h. 5erlaDaa /ea a3si as4iri a irreCersiel8 NSAI$ laia se4erti i-4r7Ce ata- i/7metasi meea3a 4ehamata terha/a4 ,OB ai3 reCersiel ma-4- irreCersiel melal-i 37m4etisi /ea s-strat8 ait- asam ara3hi/7at.
.1.&. $lasi%ikasi NSA#D
1. '-r-a asam salisilat: • • •
As4iri Salisilami/ $ifl-isal
As4iri a/alah ae atiiflamasi a tert-a8 mer-4a3a 4ehamat 4r7stala/i a me-r-3a 4r7ses iflamasi /a /ah-l- mer-4a3a ae atiiflamasi a 4ali seri /i4a3ai seal-m a/aa i-4r7fe. As4iri a /ea /7sis tii -t-3 iflamasi meea3a rasa ti/a3 ea3 4a/a lam-.a/a sit-asi se4erti ii8 iasaa /i-a3a talet eteri>;>7ate/. As4iri ti/a3 7leh /i4a3ai ersama;sama /ea NSAIANSAI$ 3area me-r-3a 3a/ar NSAIANSAI$ /alam /arah /a
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