EFECTOS ADRENERGICOS DIRECTOS.
EFECTOR
RESPUESTA
OJO -Fibras radiales músculo
contracción ( α1) => midriasis
esfínter iris -Músculo ciliar -Presión intraocular
relajación (β2) aumenta
CORAZON ( 1) - Nódulo sinusal -Aurícula -
Nódulo A-V
-Ventrículos
aumento frecuencia cardiaca Aumento contractilidad y velocidad de conducción aumento velocidad de conducción aumento contractilidad, velocidad de conducción y automatismo.
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EFECTOS ADRENERGICOS DIRECTOS.
EFECTOR
RESPUESTA
VASOS SANGUINEOS -Arterias piel, mucosas, esplácnico vasoconstricción (α1) -Arterias músculo esquelético vasocontricción (α1) vasodilatación (β2) -Arterias cerebrales vasoconstricción (α1) -Arterias coronarias vasoconstricción (α1) vasodilatación (β2) Venas vasoconstricción (α1)
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EFECTOS ADRENERGICOS DIRECTOS.
EFECTOR
RESPUESTA
TRACTO G.I. -Tono y motilidad
disminución (α, β)
-Secreciones -Esfínteres
-------------contracción (α1)
VESICULA BILIAR Y
relajación (β2)
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EFECTOS ADRENERGICOS DIRECTOS.
EFECTOR
RESPUESTA
ORGANOS SEXUALES MASCULINOS -Organos sexuales masculinos eyaculación (α1) SECRECIONES ( 1) Glándulas sudoríparas -Glándulas lagrimales
aumento secreción (localizada) aumento secreción
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EFECTOS ADRENERGICOS DIRECTOS.
EFECTOR
RESPUESTA
APARATO
estimulación renina (β1,β2)
YUXTAGLOMERULAR
inhibición renina (α2)
METABOLISMO -Hígado
glicogenolisis (α1)
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FUNCIONES ASOCIADAS CON RECEPTORES ADRENERGICOS. RECEPTORES ALFA VASOCONSTRICCION (mucosa, cutánea, esplácnica). CONTRACCION CAPSULA ESPLENICA. CONTRACCION MUSCULOS PILOMOTORES. CONTRACCION FIBRAS RADIALES MUSCULO ESFINTER DEL IRIS. CONTRACCION ESFINTERES GASTROINTESTINALES. AUMENTO SECRECION SALIVAL. RELAJACION INTESTINAL .
RECEPTORES BETA. VASODILATACION (musculatura esquelética). RELAJACION BRONQUIAL. RELAJACION LEVE MUSCULO CILIAR . RELAJACION INTESTINAL. C RONOTROPIA POSITIVA INOTROPIA POSITIVA. BATMOTROPIA POSITIVA. GLICOGENOLISIS. AUMENTO LACTICEMIA. LIPOLISIS.
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Fibra adrenérgica e intervención farmacológica
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FARMACOS QUE AUMENTAN ACTIVIDAD ADRENERGICA. De acción en la fibra adrenérgica: 2. Apor Aporte te de prec precur ursor sores es:: Dop Dopam amin ina, a, L-Do L-Dopa pa..
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FARMACOS QUE DISMINUYEN ACTIVIDAD ADRENERGICA. De acción en la fibra adrenérgica: 2. Inhibi Inhibició ciónn de de enzi enzima mass que que part partici icipan pan en la sínte síntesis sis:: Alfa-metil-para-tirosina.
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FARMACOS QUE DISMINUYEN ACTIVIDAD ADRENERGICA.
Efectos laterales comunes : Hipotensión postural
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TIPO DE RECEPTORES ADRENERGICOS
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FARMACOS ANTIADRENERGICOS ANTAGONISTAS REVERSIBLES YOHIMBINA
2
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FARMACOS ANTIADRENERGICOS ANTAGONISTAS 1y 1y 2 BLOQUEO REVERSIBLE BLOQUEO RECAPTACION N.A. AGONISTA PARCIAL β 2
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Hipertensión Arterial
Fármacos antihipertensivos 2. Simpaticolíticos: Bloqueadores beta •Bloqueadores beta inespecíficos: Propranolol. • Bloqueadores beta inespecíficos con actividad agonista :
Pindolol, Oxprenolol. Bloqueadores cardioselectivos: Metoprolol, Atenolol, Esmolol. Bloqueadores cardioselectivos con actividad agonista :
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FARMACOS ANTIADRENERGICOS ANTAGONISTAS NO SELECTIVOS PROPRANOLOL ALPRENOLOL, NADOLOL, TIMOLOL, SOTALOL.
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FARMACOS ANTIADRENERGICOS ANTAGONISTAS 1 METOPROLOL, ATENOLOL, ESMOLOL. ANTAGONISTAS 1 CON ACTIVIDAD AGONISTA AGONISTA ACEBUTOLOL, PENBUTOLOL. ANTAGONISTAS 1 CON ACTIVIDAD AGONISTA CELIPROLOL, DILEVALOL
1 1y 2
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FARMACOS ANTIADRENERGICOS β
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PRINCIPALES EFECTOS DE ESTIMULANTES GANGLIONARES. SITIO
TONO PREDOMINANTE
EFECTO
ARTERIOLAS
SIMPATICO
vasoconstricción, disminución del flujo periférico, hipertensión.
VENAS
SIMPATICO
contracción, aumento del retorno venoso y aumento del débito cardíaco.
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Trusted by over 1 million members
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Trusted by over 1 million members
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PRINCIPALES EFECTOS DE BLOQUEADORES GANGLIONARES. SITIO
TONO PREDOMINANTE
EFECTO DEL BLOQUEO
ARTERIOLAS
SIMPATICO
vasodilatación, aumento del flujo periférico, hipotensión
VENAS
SIMPATICO
dilatación, éstasis, disminución del retorno venoso y disminución del débito cardíaco.