BIPERIDENO NOMBRE COMERCIAL: PRESENTACION: MECANISMOS DE ACCION: INDICACIONES: CONTRAINDICACIONES: EFECTOS ADVERSOS: POSOLOGIA: CUIDADOS DE ENFERMERIA:
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Nombre Genérico
Biperideno Nombre Comercial
Akinetón; Bero!n Grupo
PSI"UIATR#A $ NEUROLOG#A Subgrupo
ANTIPAR%INSONIANOS Comentario de Acción Terapéutica
Se p&ede &'(r p(r( p(rkin'oni')o ind&*ido por )edi*()ento'+ Dosis
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Midri('i'2 'e?&ed(d @&*(.2 *on'tip(*ión2 reten*ión &rin(ri(2 *on&'ión )ent(.2 di't&r@io' en e. *o)port()iento2 'o)no.en*i(+ ipoten'ión t(?&i*(rdi( d&r(nte de'p&' de .( (d)ini'tr(*ión E+V++ Forma de resentación
Co)pri)ido': )4 Ret(rd: 3 )4 A)po..(': )45). !bservación
M(neo e-*.&'io de. e'pe*i(.i't(+ Por !( E+V+ (d)ini'tr(r en or)( .ent(+ Nombre Genérico
Biperideno Nombre Comercial
Akinetón Grupo
MEDICAMENTOS UTILIADOS EN INTOICACIONES Comentario de Acción Terapéutica
Into-i*(*ión *on dro4(' ?&e prod&*en ee*to' e-tr(pir()id(.e': ne&ro.pti*o'2 )eto*.opr()id(+
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Forma de resentación
A)po..(': )45). FIN DEL LISTADO / re4i'tro'0 9 IMPRIMIR LISTADO
AKINETON ® / AKINETON RETARD ARMSTRONG Denominación genérica: Biperideno. Forma farmacéutica formu!ación: Tabletas. Cada tableta contiene: clorhidrato de biperideno 2 mg. Excipiente cbp 1 tableta. Tabletas de liberación prolongada. Cada tableta contiene: clorhidrato de biperideno 4 mg. Excipiente cbp 1 tableta. Solución inyectable: cada ampolleta contiene: lactato de biperideno mg !e"ui#alente a $.% mg. de biperideno&. 'gua inyectable cbp 1 ml. biperi ride deno no est( est( indi indica cado do para para:: en)e en)erm rmed edad ad de *ar+ *ar+in inso son n y s,nd s,ndro rome mes s In"icacione# In"icacione# tera$éutica#: tera$éutica#: El bipe par+insonianos- especialmente para contrarrestar la rigide muscular y el temblor. S,ntomas extrapiramidales como diston,a aguda- acatisia y s,ndrome par+insoniano inducido por neurol/pticos y medicamentos de acción similar- en especial: haloperidol- tioridaina- tri)luoroperaina- per)enaina- etc. En#enenamiento con nicotina y con compuestos
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re#ersible re#ersible a los receptores de acetilcolina. acetilcolina. *ueden minimiarse minimiarse los s,ntomas s,ntomas como la hipersali#ación hipersali#ación o el aumento de la sudorac sudoración ión con el biperid biperideno. eno. *or tanto tanto tambi/ tambi/n n se recomienda recomienda como terapia terapia aditi#a aditi#a a la le#odop le#odopa a o medi medica camen mento tos s simil similar ares es-- "ue "ue tiene tienen n un mayor mayor e)ecto e)ecto sobre sobre la acin acinesi esia a en los los pacie paciente ntes s con con par+i par+inso nson. n. Propiedades farmacodinámic farmacodinámicas: as: mecanismo mecanismo de acción: acción: el biperideno es un Farmacocinética farmaco"inamia: Propiedades agente anticolin/rgico con un marcado e)ecto sobre sistema ner#ioso central. En comparación con la atropina- tiene e)ectos anticolin/rgicos d/biles. os estudios sobre la unión a los receptores muscar,nicos humanos muestran una alta alta a)inida a)inidad d del biperiden biperideno o por la subclas subclase e 1- el princip principal al tipo tipo de recept receptor or muscar, muscar,nic nico o en el cerebr cerebro. o. a administració administración n de biperideno tiene una in)luencia in)luencia )a#orable en el temblor causado por los agentes agentes colin/rgicos colin/rgicos con acti#idad central !tremorina- pilocarpina& o la catalepsia y rigide muscular producidas por la administración de neurol/pticos o reserpina en animales. Se ha demostrado un e)ecto acti#ador psicomotor del biperideno en #arios modelos animales. Propiedades farmacocinéticas: despu/s farmacocinéticas: despu/s de la administración oral- el clorhidrato de biperideno !4 mg "ue corresponden a $-3 mg de biperideno& biperideno& se absorbe r(pidamente r(pidamente con un retraso de media hora y tiene una #ida media de -$ horas. Se alcanan alcanan las concentraciones concentraciones plasm(ticas plasm(ticas pico de aproximadamente aproximadamente 4 ng5ml despu/s de aproximadamente 1. horas. El #olumen de distribución aparente es de 24 6 4-1 litros5+g. a tasa de aclaramiento plasm(tico oral es alrededor de 147 litros5hora8 la biodisponibilidad es aproximadamente del $$9 y la #ida media de eliminación de 21 horas. espu/s una dosis oral ;nica de biperideno 4 mg- la #ida media de eliminación terminal en
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comparación con la tableta de liberación instant(nea- la absorción de la presentación de liberación prolongada se retrasa considerablemente- con un primer pico de concentración plasm(tica a las $- horas y un segundo pico de 1ng5ml 1ng5ml despu/s despu/s de 1 a 12 horas. a #ida #ida media media terminal terminal dura dura aproxim aproximadam adamente ente 24 horas horas despu/s despu/s de la administración de la presentación de liberación prolongada. a biodisponibilidad es aproximadamente la misma para las dos presentaciones orales. El biperideno se une de )orma importante a las prote,nas plasm(ticas. 'dem(s de la alb;min alb;minaa- un )i0ado )i0adorr potenci potencial al es la α1= glucopr glucoprote, ote,na na (cida (cida !α1 '>*&. El porcenta0e de la unión- el cual es indepen independien diente te de la concent concentrac ración ión hasta hasta alcanar alcanar una cantida cantidad d mucho mucho mayor mayor "ue el ni#el ni#el terap/u terap/utic ticoo- es aproximadamente de 39 en los cauc(sicos y aproximadamente 39 en los 0aponeses. ?o se sabe la causa de esta di)erencia. di)erencia. El biperideno se une a las prote,nas plasm(ticas plasm(ticas un 349 en las mu0eres y un 3$9 en los hombres. El biperideno se metabolia casi completamente. ?o se detecta biperideno sin cambios en la orina. El principal metabolito del biperideno se )orma por hidroxilación del anillo bicicloheptano !79&- aun"ue tambi/n se produce algo de hidroxilación en el anillo piperidina !49&. 'proximadamente cantidades iguales de #arios metabolitos !productos de hidroxilación y con0ugados& se excretan por la orina y las heces. ?o existen estudios del metabolismo del biperideno despu/s de administración intra#enosa. ?o existe in)ormación disponible acerca de la )armacocin/tica en pacientes con alteraciones de la )unción hep(tica y renal. %ontrain"icacione#: El biperideno est( contraindicado en: hipersensibilidad a la sustancia acti#a o a alguno de los
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e#itarse el consumo de alcohol. Embarazo: no se sabe si el biperideno puede causar Re#triccione# "e u#o "urante e! em'ara(o !a !actancia: Embarazo: no daAo )etal cuando se administra a mu0eres embaraadas o si puede a)ectar la capacidad de reproducción. ebe administrarse el biperideno en mu0eres embaraadas sólo si es claramente necesario. Lactancia: no se sabe si se excreta el biperideno en la leche humana. Como muchos medicamentos se excretan en la leche humana- debe tenerse precaución cuando se administra el biperideno a una mu0er lactando. Reaccio Reaccio post rcializ rcializaci ación ón estudio estudio clínic clínic list list Reaccio Reaccio n"aria# n"aria# a")
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e)ectos secundarios del sistema ner#ioso central y peri)/rico pueden alterar la capacidad para mane0ar y operar ma"uinaria. a administración concomitante de "uinidina puede aumentar el e)ecto de /sta y disminuir la conducción en el nodo '. a experiencia del uso de biperideno- en tabletas y ampolletas en los niAos- se limita a su empleo tran transi sito torio rio para para corr corregi egirr las las dist diston, on,as as pro# pro#oca ocada das s por por medic medicam ament entos os-- prin princip cipal almen mente te los los neur neurol/ ol/pt ptico icos. s. A!teracione# en !o# re#u!ta"o# "e $rue'a# "e !a'oratorio: ?o se han demostrado alteraciones en las pruebas de laboratorio con el uso agudo o crónico de biperideno- excepto con la administración intra#enosa para la "ue se report ligera y transitoria disminución disminución del cortisol cortisol plasm(tico y de la prolactina. os par(metros cl,nico
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eriátrico: se debe debe tene tenerr preca precauci ución ón al dosi) dosi)ic icar ar y admin adminis istr trar ar biper biperid iden eno o en pacie paciente ntes s de edad edad a#an a#anad adaaespecialmente en a"u/llos con s,ntomas de en)ermedad org(nica cerebral y en pacientes con susceptibilidad increme incrementa ntada da a crisis crisis cerebra cerebrales. les. os paciente pacientes s de edad a#anada a#anada son m(s sensibl sensibles es a los medicame medicamento ntos s anticolin/rgicos. "(I)ET*) anticolin/rgicos. "(I)ET*) Retard+ tabletas de , m: es adecuado para a"uellos pacientes en los "ue- por alguna indicación especial y con necesidades de dosis altas- se desee disminuir el n;mero de tomas diarias. a dosis promedio en el adulto es de 1 a 2 tabletas al d,a y como m(ximo- $ tabletas al d,a- repartidas e"uitati#amente en 24 h. "(I)ET*) h. "(I)ET*) solución in!ectable: adultos: biperideno solución inyectable mg5ml es especialmente ;til en los
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lactato de biperideno para inyección en )orma repetida por #,a intra#enosa hasta "ue se resuel#an los s,ntomas de intoxicación. 'so eriátrico: Se re"uiere precaución al dosi)icar a los pacientes mayores- especialmente a"uellos con s,ntomas de en)ermedad org(nica cerebral y pacientes con una susceptibilidad aumentada a las crisis con#ulsi#as. os pacientes mayores son m(s sensibles a los medicamentos anticolin/rgicos. 'so pediátrico: Trastornos motores inducidos inducidos por medicamentos: medicamentos: Es limitad limitada a la experie experiencia ncia del uso pedi(tr pedi(trico ico del biperid biperideno eno y princi principal palment mente e se relaci relaciona ona a tratam tratamien ientos tos de corto corto plao plao de la diston, diston,a a induci inducida da por medica medicament mentos os !por e0emplo e0emplo causada causada por l/ ti t l id t i il &
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primaria para e#itar "ue contin;e la absorción del medicamento. Se recomienda lubricar la sonda nasog(strica debido a "ue las mucosas podr,an estar secas. Como ant,doto de elección- se recomienda la )isostigmina a dosis de 1 mg !- mg en niAos y ancianos& por #,a intramuscular o intra#enosa lenta- pudi/ndose repetir una segunda aplicación a los 2 min8 si no se obtu#o me0or,a- hasta un m(ximo total de 4 mg !en niAos y ancianos- 2 mg&. El tratamiento de la sobredosi)icación incluye las medidas generales de mantenimiento- como asegurar las #,as a/reas permeab permeables les-- admini administra stración ción de ox,geno ox,geno-- mantene mantenerr permeab permeable le una #,a endo#en endo#enosaosa- uso de sonda sonda #esical #esical-)ortalecimien )ortalecimiento to de la )unción card,ac !aplicación !aplicación de sores& y control con medios ),sicos la hipertermia- si
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